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A ranar 15 ga Afrilu, 2022, an kammala samar da matukin jirgi na Lecardipine hydrochloride babban zobe a lokaci guda, kuma ƙarfin samarwa na yanzu shine 5Mt/ wata.

A ranar 15 ga Afrilu, 2022, an kammala samar da matukin jirgi na Lecardipine hydrochloride babban zobe a lokaci guda, kuma ƙarfin samarwa na yanzu shine 5Mt/ wata.
Sunan Ingilishi:Lercanidipine hydrochloride
Sunan sinadarai:1,4-Dihydro-2,6-dimethyl-4- (3-nitrophenyl) -3,5-pyridinedicarboxylic acid 2-[(3,3-di phenylpropyl) methylamino] -l, l-dimethylethyl methyl ester hydrochloride.

Lambar CAS: 132866-11-6
Aikace-aikace:Don kula da maganin Lecardipine hydrochloride, ba zai yi mummunan tasiri akan glucose na jini da matakan lipid ba, kuma yana da tasirin antihypertensive mai ƙarfi.

Hasashen kasuwa:
Akwai mutane sama da miliyan 200 da ke fama da cutar hawan jini a kasar Sin, kuma ana samun sabbin masu kamuwa da cutar hawan jini miliyan 10 a kowace shekara, yawancinsu ba a kula da su ba, lamarin da ke haddasa yawaitar matsalolin hauhawar jini kamar shanyewar jiki, da mace-mace a kasar Sin a duk shekara a cikin 3. miliyan masu fama da cututtukan zuciya, 50% suna da alaƙa da hauhawar jini, kuma farashin jiyya na cututtukan zuciya ya kai yuan biliyan 309.8 kowace shekara.Dalilin rashin kula da marasa lafiya ba wai kawai ya kamata a inganta fahimtar marasa lafiya game da hauhawar jini da matsalolinsa ba, har ma da yawancin marasa lafiya da ke buƙatar shan magungunan rayuwa ba su da kyau kuma ba za su iya shan magani a kowace rana ba, amma wannan kuma ya nuna cewa. Kasuwar magungunan antihypertensive tana da yuwuwar haɓakawa.Idan aka kwatanta da irin waɗannan kwayoyi, locarbodipine hydrochloride yana da ƙarfin zaɓi na jijiyoyin jini.Kayan sa na musamman na lipophilic yana sa shi jinkiri kuma yana dawwama yana tasirin antihypertensive Tasirin atherogenic, musamman dacewa ga masu fama da hauhawar jini tare da atherosclerosis, yana da ƙimar aikace-aikacen asibiti mai girma da fa'idar kasuwa.

Ayyukan Pharmacological:
Lecardipine wani sabon ƙarni na dihydropyridine calcium tashar tashar hysteresis wakili, tare da karfi na jijiyoyin bugun gini zažužžukan, m sakamako, karfi antihypertensive sakamako, dogon mataki lokaci, m inotropic sakamako da sauransu.Nazarin in vitro sun gano cewa locarbodipine yana da tasirin shakatawa kai tsaye a kan tsoka mai santsi na jijiyoyin jini, sabili da haka yana da tasirin antihypertensive mai ƙarfi a cikin vivo, amma yana da ɗan tasiri akan bugun zuciya da fitarwar zuciya.Saboda babban kwayar halittar hydrophobic da karfi mai solubility, locarbodipine yana da sauri rarraba zuwa kyallen takarda da gabobin bayan shiga cikin jiki, yana ɗaure da jijiyoyi masu santsi na ƙwayar tsoka, kuma yana sakewa a hankali.Sabili da haka, ko da yake maganin maganin wannan magani yana da ɗan gajeren lokaci na kawar da rashin gazawar, sakamakonsa yana da tsayi.


Lokacin aikawa: Afrilu-15-2022